First total synthesis of papilistatin.

نویسندگان

  • Meng Wu
  • Ling Li
  • An-Zheng Feng
  • Bo Su
  • De-min Liang
  • Yu-xiu Liu
  • Qing-min Wang
چکیده

Papilistatin has been isolated recently and found to have good anticancer and antibacterial activity. Papilistatin is a unique phenanthrene-1,10-dicarboxylic acid. The first total synthesis of papilistatin is described here with radical cyclisation as the key step.

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عنوان ژورنال:
  • Organic & biomolecular chemistry

دوره 9 7  شماره 

صفحات  -

تاریخ انتشار 2011